Affinity DataIC50: 112nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
Affinity DataEC50: 549nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair