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Found
1
Enz. Inhib. hit(s) with Target = 'Estrogen receptor [298-554]' and Ligand = 'BDBM521378'
Target
Estrogen receptor [298-554]
(Homo sapiens (Human))
Sanofi
US Patent
Ligand
BDBM521378
(5-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)
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Affinity Data
IC50: 1nM
Assay Description:
Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...
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Target Info
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Ligand Info
PC cid
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Details
US Patent
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