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Found 2 Enz. Inhib. hit(s) with Target = 'Estrogen receptor beta' and Ligand = 'BDBM50223229'
TargetEstrogen receptor beta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50223229((8R,9S,10R,13S,14S,17S)-3,10,13-trimethyl-2,7,8,9,...)
Affinity DataIC50:  9.40nMAssay Description:Binding affinity at human recombinant ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50223229((8R,9S,10R,13S,14S,17S)-3,10,13-trimethyl-2,7,8,9,...)
Affinity DataEC50:  220nMAssay Description:Agonist activity at ERbeta expressed in HEK293 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed