Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Extracellular calcium-sensing receptor' and Ligand = 'BDBM50299678'
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50299678((1R)-2-methyl-N-((1R)-1-phenylethyl)-1-(1-(4-(trif...)
Affinity DataEC50:  2.34E+3nMAssay Description:Activity at human CaSR expressed in HEK293 cells assessed as calcium release by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed