Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Fatty-acid amide hydrolase 1' and Ligand = 'BDBM50307083'
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Indian Institute Of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50307083(4-nitrophenyl 4-(3-phenoxybenzyl)piperazine-1-carb...)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant human FAAH incubated for 5 mins followed by substrate addition by cayman fluorescence based multimode microplate reader ass...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Indian Institute Of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50307083(4-nitrophenyl 4-(3-phenoxybenzyl)piperazine-1-carb...)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant FAAH (unknown origin) expressed in COS7 cells assessed as blockade of substrate hydrolysis using 2-AG as substrate preincub...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50307083(4-nitrophenyl 4-(3-phenoxybenzyl)piperazine-1-carb...)
Affinity DataIC50:  13nMAssay Description:Inhibition of FAAH in mouse brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Indian Institute Of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50307083(4-nitrophenyl 4-(3-phenoxybenzyl)piperazine-1-carb...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated with enzyme for 10 mins followed by substrate addition for 2 hrs by fluor...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Indian Institute Of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50307083(4-nitrophenyl 4-(3-phenoxybenzyl)piperazine-1-carb...)
Affinity DataIC50:  40nMAssay Description:FAAH inhibition assay was performed using Fatty Acid Amide Hydrolase Inhibitor Screening Assay Kit (Item #10005196), Cayman (1180 E Ellsworth Rd Ann ...More data for this Ligand-Target Pair
In DepthDetails US Patent