Found 33 Enz. Inhib. hit(s) with Target = 'Fatty-acid amide hydrolase 1 [30-579]' and Ligand = 'BDBM26739' 
Affinity DataKi: 2.00E+3nMAssay Description:Enzyme-coupled assay using oleamide as substrate where stoichiometic quantites of NAD are formed upon the generation of ammonia from oleamide by FAAH...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FAAH in Wistar rat brain intact neurons assessed as reduction in [3H]anandamide hydrolysis using [3H]anandamide as substrate preincubat...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of rat intact neuron FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenates preincubated for 10 mins followed by addition of substrate measured after 30 mins by liqui...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of rat FAAH assessed as hydrolysis of anandamidoaminomethylcumarinMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of FAAH in Wistar rat cerebral membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.57nMAssay Description:Displacement of [3H]-anandamide from rat brain FAAH after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Displacement of [3H]anandamide from FAAH in rat brain membranes after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of FAAH in Wistar rat brain membranes using [3H]-anandamide as substrate preincubated for 10 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of FAAH in rat brain membrane using anandamide[ethanolamine-3H] as substrate assessed as reduction in [3H]-ethanolamine production incubat...More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of FAAH in Wistar rat brain membranes assessed as reduction in [3H]anandamide hydrolysis using [3H]anandamide as substrate preincubated fo...More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of FAAH in rat brain membrane assessed as [3H]anandamide hydrolysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of [3H]-anandamide binding to fatty acid amide hydrolase of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of rat brain membrane FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Inhibition of rat histidine tagged FAAH expressed in Escherichia coli by coumarin ester substrate fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of FAAH in rat brain membranes assessed as hydrolysis of [14C]-anandamide preincubated for 20 mins before [14C]-anandamide addition measur...More data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:The assays for compounds described herein are amenable to high throughput screening. Preferred assays thus detect binding of the inhibitor to FAAH or...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of FAAH in rat brain microsomes using OMP substrate by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate preincubated for 10 mins at pH 8More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of rat FAAH incubated 3 hrs prior to addition of arachidonylaminomethylcoumarin amideMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMpH: 9.0Assay Description:Inhibition of FAAH in rat brain membrane at pH 9 using N-arachidonoyl-[14C]-ethanolamine as substrate preincubated for 10 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of FAAH in rat brain membrane using N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide as substrate measured after 60 mins by reverse-phase HPLC-ba...More data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of rat FAAH preincubated for 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of FAAH in rat brain microsomes using N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide as substrate after 60 mins by fluorescence-based HPLC anal...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of FAAH in rat brain microsomes using N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide as substrate after 60 mins by fluorescence-based reversed ...More data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain microsomes assessed as N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide conversion to 4-pyren-1-ylbutanoic ac...More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of rat FAAH incubated 1 hr prior to addition of arachidonylaminomethylcoumarin amideMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate preincubated for 10 mins at pH 6More data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Inhibition of Sprague-Dawley rat brain microsome FAAH assessed as reduction in 4-pyren-1-ylbutanoic acid release after 60 mins by reverse phase HPLC-...More data for this Ligand-Target Pair
Affinity DataIC50: 141nMpH: 7.4Assay Description:Inhibition of FAAH in rat brain membrane at pH 7.4 using N-arachidonoyl-[14C]-ethanolamine as substrate preincubated for 10 mins followed by substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of FAAH from rat brain microsomes by RP-HPLCMore data for this Ligand-Target Pair
