Found 4 Enz. Inhib. hit(s) with Target = 'Fatty-acid amide hydrolase 1 [30-579]' and Ligand = 'BDBM97458'
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 90 mins prior to ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 9.40nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 45 mins prior to ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of FAAH in Wistar rat brain membranes using [3H]-anandamide as substrate preincubated for 10 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Membrane fractions were prepared from Wistar rat brain homogenates, and FAAH activity were assayed by using [3H]anandamide (anandamide[ethanolamine-3...More data for this Ligand-Target Pair