Affinity DataIC50: 45nMAssay Description:Inhibition of FAK (unknown origin) using biotinylated His-TEV-hsFAK(31-686)(K454R) substrate after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Inhibition of FAK in human HT-29 cells assessed as phosphorylation at tyrosine 397 after 45 minsMore data for this Ligand-Target Pair
Affinity DataKd: 35nMAssay Description:Binding affinity to FAK (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair