Found 3 Enz. Inhib. hit(s) with Target = 'G protein-coupled receptor kinase 4' and Ligand = 'BDBM2579'
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 69.9nMAssay Description:Inhibition of human GRK4 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Inhibition of human GRK4 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 37nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair