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Found 4 Enz. Inhib. hit(s) with Target = 'G protein-coupled receptor kinase 5' and Ligand = 'BDBM50529458'
TargetG protein-coupled receptor kinase 5(Bos taurus)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50529458(CHEMBL4557065)
Affinity DataIC50:  700nMAssay Description:Inhibition of bovine GRK5 C474S mutant using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor kinase 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50529458(CHEMBL4557065)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human GRK5 using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor kinase 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50529458(CHEMBL4557065)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of human GRK5 using tubulin as substrate measured after 100 mins by [gamma-32P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor kinase 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50529458(CHEMBL4557065)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human GRK5 using tubulin as substrate measured after 0 mins by [gamma-32P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed