Found 4 Enz. Inhib. hit(s) with Target = 'G-protein coupled bile acid receptor 1' and Ligand = 'BDBM50414954' 
Affinity DataEC50: 31.6nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Agonist activity at rat TGR5 expressed in melanophores assessed as melanosome dispersion by melanophore assayMore data for this Ligand-Target Pair
Affinity DataEC50: 31.6nMAssay Description:Agonist activity at human TGR5 expressed in melanophores assessed as melanosome dispersion by melanophore assayMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at TGR5 expressed in human U2-OS cells assessed as increase in MRE/CRE-driven gene expression by luciferase reporter gene assayMore data for this Ligand-Target Pair
