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Found 3 Enz. Inhib. hit(s) with Target = 'G-protein coupled receptor 39' and Ligand = 'BDBM50232367'
TargetG-protein coupled receptor 39(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50232367(CHEMBL4093273)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 39(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50232367(CHEMBL4093273)
Affinity DataEC50:  380nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 39(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50232367(CHEMBL4093273)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed