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Found 3 Enz. Inhib. hit(s) with Target = 'G-protein coupled receptor 52' and Ligand = 'BDBM50554930'
TargetG-protein coupled receptor 52(Homo sapiens (Human))
University Of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50554930(CHEMBL4761381 | US20240059655, Compound PW0878)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human GPR52 expressed in HEK293 cells assessed as increase in cAMP levels incubated for 15 mins by Glosensor cAMP assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Mus musculus)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM50554930(CHEMBL4761381 | US20240059655, Compound PW0878)
Affinity DataEC50:  90nMAssay Description:In Vitro Evaluation of GPR52 Activation. Newly synthesized compounds were evaluated in a twelve-point concentration-response for GPR52 agonist activi...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled receptor 52(Mus musculus)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM50554930(CHEMBL4761381 | US20240059655, Compound PW0878)
Affinity DataEC50:  90nMAssay Description:In Vitro Evaluation of GPR52 Activation. Newly synthesized compounds were evaluated in a twelve-point concentration-response for GPR52 agonist activi...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent