Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'GABA-A receptor; alpha-2/beta-3/gamma-2' and Ligand = 'BDBM50007552'
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
University Of Wisconsin-Milwaukee

Curated by ChEMBL
LigandPNGBDBM50007552(6-Methoxy-4-methoxymethyl-9H-beta-carboline-3-carb...)
Affinity DataKi:  1.19nMAssay Description:Binding affinity measured using LtK- cell membranes expressing GABA alpha2-beta3-gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
University Of Wisconsin-Milwaukee

Curated by ChEMBL
LigandPNGBDBM50007552(6-Methoxy-4-methoxymethyl-9H-beta-carboline-3-carb...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-2-beta-3-gamma-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed