Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Gag-Pol polyprotein [489-587]' and Ligand = 'BDBM1136'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM1136((4R,5R,6R)-6-benzyl-5-hydroxy-1-(1H-indazol-5-ylme...)
Affinity DataKi:  1.20nMAssay Description:Inhibitory activity of compound against HIV-1 aspartyl protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM1136((4R,5R,6R)-6-benzyl-5-hydroxy-1-(1H-indazol-5-ylme...)
Affinity DataKi:  1.20nMAssay Description:Inhibition constant of HIV protease inhibitorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM1136((4R,5R,6R)-6-benzyl-5-hydroxy-1-(1H-indazol-5-ylme...)
Affinity DataKi:  1.20nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed