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Found 4 Enz. Inhib. hit(s) with Target = 'Gag-Pol polyprotein [489-587]' and Ligand = 'BDBM50004780'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of California

Curated by ChEMBL
LigandPNGBDBM50004780(3-[18-(2-Carboxy-ethyl)-8,13-bis-(1,2-diacetoxy-et...)
Affinity DataKi:  85nMAssay Description:Binding affinity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of California

Curated by ChEMBL
LigandPNGBDBM50004780(3-[18-(2-Carboxy-ethyl)-8,13-bis-(1,2-diacetoxy-et...)
Affinity DataIC50:  100nMAssay Description:Inhibitory concentration against HIV-1 protease in the absence of DMSOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of California

Curated by ChEMBL
LigandPNGBDBM50004780(3-[18-(2-Carboxy-ethyl)-8,13-bis-(1,2-diacetoxy-et...)
Affinity DataIC50:  400nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of California

Curated by ChEMBL
LigandPNGBDBM50004780(3-[18-(2-Carboxy-ethyl)-8,13-bis-(1,2-diacetoxy-et...)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed