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Found 3 Enz. Inhib. hit(s) with Target = 'Galectin-3' and Ligand = 'BDBM541639'
TargetGalectin-3(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM541639(US11267811, Example 250)
Affinity DataIC50:  10nMAssay Description:The Gal-3 assays were performed in 384 white Opti plates in three replicates at room temperature with gentle shaking at 250-300 rpmFrom the original ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGalectin-3(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM541639(US11267811, Example 250)
Affinity DataIC50:  15nMAssay Description:Inhibition of His-tagged recombinant human Gal-3 preincubated for 30 mins followed by B-ASF addition measured after 1 hr by time resolved fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGalectin-3(Mus musculus)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM541639(US11267811, Example 250)
Affinity DataIC50:  126nMAssay Description:Inhibition of His-tagged recombinant mouse Gal-3 preincubated for 30 mins followed by B-ASF addition measured after 1 hr by time resolved fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed