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Found 2 Enz. Inhib. hit(s) with Target = 'Gamma-hydroxybutyrate receptor' and Ligand = 'BDBM50246039'
TargetGamma-hydroxybutyrate receptor(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50246039((S,E)-2-(5-hydroxy-8,9-dihydro-5H-benzo[7]annulen-...)
Affinity DataIC50:  7.40E+4nMAssay Description:Displacement of [3H]SUC from succinic acid binding site of gamma-hydroxybutyrate receptor in rat forebrain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-hydroxybutyrate receptor(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50246039((S,E)-2-(5-hydroxy-8,9-dihydro-5H-benzo[7]annulen-...)
Affinity DataIC50:  9.30E+4nMAssay Description:Displacement of [3H]GHB from gamma-hydroxybutyrate binding site of gamma-hydroxybutyrate receptor in rat forebrain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed