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Found 3 Enz. Inhib. hit(s) with Target = 'Genome polyprotein/Non-structural protein 4A' and Ligand = 'BDBM103841'
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
University Of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM103841(5172-mcP1P3)
Affinity DataKi:  2nMAssay Description:Inhibition of wild type HCV genotype 1a NS3/4A protease expressed in Escherichia coli BL21(DE3) using Ac-DE-Dap(QXL 520)-EE-Abu-psi-[COO]AS-C(5-FAMsp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
University Of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM103841(5172-mcP1P3)
Affinity DataKi:  3.10nMAssay Description:Inhibition of HCV genotype 1a NS3/4A protease R155K mutant expressed in Escherichia coli BL21(DE3) using Ac-DE-Dap(QXL 520)-EE-Abu-psi-[COO]AS-C(5-FA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
University Of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM103841(5172-mcP1P3)
Affinity DataKi:  91nMAssay Description:Inhibition of HCV genotype 1a NS3/4A protease D168A mutant expressed in Escherichia coli BL21(DE3) using Ac-DE-Dap(QXL 520)-EE-Abu-psi-[COO]AS-C(5-FA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed