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Found 4 Enz. Inhib. hit(s) with Target = 'Genome polyprotein' and Ligand = 'BDBM50026765'
TargetGenome polyprotein(West Nile virus)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50026765(CHEMBL3335494)
Affinity DataKi:  4.90E+4nMAssay Description:Inhibition of West Nile virus serotype 2 NS2B-NS3 protease by homogeneous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50026765(CHEMBL3335494)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of Dengue virus serotype 2 NS2B-NS3 protease preincubated with protein for 15 mins followed by Abz-Nle-Lys-Arg-Arg-Ser-3-(NO2)Tyr substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50026765(CHEMBL3335494)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of Dengue virus serotype 2 NS2B-NS3 protease by homogeneous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50026765(CHEMBL3335494)
Affinity DataIC50:  5.80E+4nMAssay Description:Inhibition of West Nile virus serotype 2 NS2B-NS3 protease by homogeneous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed