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Found 3 Enz. Inhib. hit(s) with Target = 'Genome polyprotein' and Ligand = 'BDBM50366760'
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50366760(CHEMBL2369589)
Affinity DataKi:  0.75nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50366760(CHEMBL2369589)
Affinity DataKi:  9nMAssay Description:Inhibition of HCV genotype-1a full length NS3 protease preincubated for 10 mins followed by Ac-DED(Edans)EEAbuj-[COO]ASK(Dabcyl)-NH2 addition in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50366760(CHEMBL2369589)
Affinity DataKi:  12nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed