Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Geranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50100277'
LigandPNGBDBM50100277(2-(3-Benzyl-phenoxy)-4-imidazol-1-ylmethyl-benzoni...)
Affinity DataIC50:  600nMAssay Description:Displacement of radiolabeled FTI from Farnesyltransferase in cultured v-Ha-ras-transformed RAT1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed