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Found 6 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Ligand = 'BDBM50265673'
TargetGlucocorticoid receptor(Homo sapiens (Human))
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50265673(CHEMBL4068611)
Affinity DataKi:  7.20nMAssay Description:Antagonist activity at glucocorticoid receptor in human HepG2 cells assessed as inhibition of dexamethasone-induced tyrosine amino transferase activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50265673(CHEMBL4068611)
Affinity DataKi:  12nMAssay Description:Antagonist activity at rat glucocorticoid receptor in primary hepatocytes assessed as dexamethasone-induced tyrosine amino transferase activity prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50265673(CHEMBL4068611)
Affinity DataKi:  81nMAssay Description:Antagonist activity at glucocorticoid receptor in human primary hepatocytes assessed as inhibition of dexamethasone-induced tyrosine amino transferas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Canis lupus familiaris)
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50265673(CHEMBL4068611)
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at dog glucocorticoid receptor in primary hepatocytes assessed as dexamethasone-induced tyrosine amino transferase activity prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50265673(CHEMBL4068611)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat glucocorticoid receptor in primary hepatocytes assessed as induction of tyrosine amino transferase activity measured after 20...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Canis lupus familiaris)
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50265673(CHEMBL4068611)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at dog glucocorticoid receptor in primary hepatocytes assessed as induction of tyrosine amino transferase activity measured after 20...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed