Affinity DataKi: 108nMAssay Description:Displacement of [3H]AMPA from GluA2-S1S2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 348nMAssay Description:Displacement of [3H[AMPA from rat recombinant GluA2(R)o expressed in sS9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.46E+4nMAssay Description:Agonist activity at rat recombinant GluA2(Q)i expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair