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Found 3 Enz. Inhib. hit(s) with Target = 'Glutamate receptor 2' and Ligand = 'BDBM50512944'
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512944(CHEMBL4529665)
Affinity DataKi:  320nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2-ABD expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512944(CHEMBL4529665)
Affinity DataKi:  710nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512944(CHEMBL4529665)
Affinity DataEC50:  6.50E+4nMAssay Description:Agonist activity at rat GluA2(Q) receptor expressed in Xenopus laevis oocytes assessed as induction of (S)-glutamate-induced channel current at -60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB