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Found 2 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, NMDA 1/2A' and Ligand = 'BDBM50164544'
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50164544((2R,3S)-1-(Biphenyl-4-sulfonyl)-piperazine-2,3-dic...)
Affinity DataKi:  1.36E+4nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50164544((2R,3S)-1-(Biphenyl-4-sulfonyl)-piperazine-2,3-dic...)
Affinity DataKi:  1.36E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed