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Found 5 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, NMDA 2B' and Ligand = 'BDBM50385169'
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50385169(CHEMBL2036513)
Affinity DataKd:  15.2nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain thalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50385169(CHEMBL2036513)
Affinity DataKd:  5.90nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain olfactory tubercleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50385169(CHEMBL2036513)
Affinity DataKd:  9.10nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50385169(CHEMBL2036513)
Affinity DataKd:  9.80nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50385169(CHEMBL2036513)
Affinity DataKd:  9.30nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain straitumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed