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Found 1 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, kainate 1' and Ligand = 'BDBM50178141'
TargetGlutamate receptor ionotropic, kainate 1(RAT)
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Curated by ChEMBL
LigandPNGBDBM50178141((S)-1-(2-amino-2-carboxyethyl)-3-(4-carboxybenzyl)...)
Affinity DataKd:  9.25E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed