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Found 3 Enz. Inhib. hit(s) with Target = 'Glycine receptor subunit alpha-1/beta' and Ligand = 'BDBM50232890'
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)
Affinity DataIC50:  56nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)
Affinity DataIC50:  210nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)
Affinity DataIC50:  214nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed