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Found 3 Enz. Inhib. hit(s) with Target = 'Glycogen phosphorylase, liver form' and Ligand = 'BDBM50136437'
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136437(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1,2,3,...)
Affinity DataIC50:  44nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136437(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1,2,3,...)
Affinity DataIC50:  44nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136437(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1,2,3,...)
Affinity DataIC50:  86nMAssay Description:Inhibition of recombinant human liver GPa by multienzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed