Found 4 Enz. Inhib. hit(s) with Target = 'Gonadotropin-releasing hormone receptor' and Ligand = 'BDBM50102450'
Affinity DataIC50: 0.580nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells as inhibition of GnRH-induced LH secretion by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.64nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.631nMAssay Description:Competitive antagonism of GnRH-induced response in the reporter gene assayMore data for this Ligand-Target Pair