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Found 4 Enz. Inhib. hit(s) with Target = 'Gonadotropin-releasing hormone receptor' and Ligand = 'BDBM50422274'
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50422274(GONADORELIN | Human gonadoliberin-i)
Affinity DataIC50:  2nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50422274(GONADORELIN | Human gonadoliberin-i)
Affinity DataIC50:  6nMAssay Description:The compound was tested for the concentration to inhibit 50% of [125 I]leuprorelin binding to Leutinizing releasing hormone receptor the membrane fra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50422274(GONADORELIN | Human gonadoliberin-i)
Affinity DataIC50:  7nMAssay Description:The compound was tested for the concentration to inhibit 50% of [125 I]leuprorelin binding to Leutinizing releasing hormone receptor in the membrane ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50422274(GONADORELIN | Human gonadoliberin-i)
Affinity DataIC50:  10nMAssay Description:The Compound was tested for the concentration to inhibit 50% of [125 I ]leuprorelin binding to the cloned human Leutinizing releasing hormone recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed