Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Gonadotropin-releasing hormone receptor' and Ligand = 'BDBM50533946'
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533946(CHEMBL4474116)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533946(CHEMBL4474116)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity against human GnRH receptor expressed in HEK293 cells co-transfected with pGL4-NFAT promoter AP1-luc assessed as inhibition of 20...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed