Found 3 Enz. Inhib. hit(s) with Target = 'Growth hormone secretagogue receptor type 1' and Ligand = 'BDBM50208662'
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cellsMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cellsMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataIC50: 275nMAssay Description:Antagonist activity at human GHSR1a receptor expressed in CHO cells assessed as reduction of ghrelin-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair