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Found 4 Enz. Inhib. hit(s) with Target = 'Growth hormone secretagogue receptor type 1' and Ligand = 'BDBM50260268'
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50260268(CHEMBL501261 | rPKPfQwFwLL-NH2)
Affinity DataKi:  77nMAssay Description:Displacement of [125I]-His9 ghrelin from SNAP-tagged human GHSR expressed in HEK293T cells after 3 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50260268(CHEMBL501261 | rPKPfQwFwLL-NH2)
Affinity DataIC50:  3.20nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50260268(CHEMBL501261 | rPKPfQwFwLL-NH2)
Affinity DataIC50:  18nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50260268(CHEMBL501261 | rPKPfQwFwLL-NH2)
Affinity DataEC50:  99nMAssay Description:Inverse agonist activity at SNAP-tagged human GHSR expressed in HEK293T cells assessed as reduction in inositol phosphate production after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed