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Found 1 Enz. Inhib. hit(s) with Target = 'HTH-type transcriptional regulator ExsA' and Ligand = 'BDBM50319089'
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319089((E)-2-(2-(4-(3-(6-acetylpyridin-3-yl)acrylamido)ph...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed