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Found 3 Enz. Inhib. hit(s) with Target = 'Heat shock protein HSP 90-alpha/90-beta' and Ligand = 'BDBM50150178'
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Conforma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50150178(CHEMBL435016 | Carbamic acid (4E,6Z,10E)-(8S,9S,12...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human epidermal growth factor 2 (Her-2) degredation in MCF-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Conforma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50150178(CHEMBL435016 | Carbamic acid (4E,6Z,10E)-(8S,9S,12...)
Affinity DataIC50:  1.20E+3nMAssay Description:Concentration required to inhbit Bis-ANS activity by recombinant heat shock protein 90 (rHSP90) conformational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Conforma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50150178(CHEMBL435016 | Carbamic acid (4E,6Z,10E)-(8S,9S,12...)
Affinity DataIC50:  3.00E+3nMAssay Description:Concentration required to inhibit biotin-GM binding to recombinant heat shock protein 90(rHsp90)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed