Affinity DataIC50: 19nMAssay Description:Binding affinity to Hsp90alpha N-terminal ATPase domain by TR-FRET assay based competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:Inhibition of Hsp90alpha ATPase activity by malachite green ATP-ase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 350nMAssay Description:Inhibition of Hsp90alpha in human SKBR3 cells assessed as ErbB2 degradation by Western blot analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Inhibition of Hsp90alpha in human H1299 cells assessed as HIF-1alpha degradation by luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Inhibition of Hsp90alpha in human SKBR3 cells assessed as up-regulation of HSP70 protein by Western blot analysisMore data for this Ligand-Target Pair