Affinity DataIC50: 9.36E+3nMAssay Description:Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
Affinity DataKd: 5.12E+3nMAssay Description:Binding affinity to recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as dissociation constant measured after 15 mins by microsc...More data for this Ligand-Target Pair