Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H1 receptor' and Ligand = 'BDBM255474'
TargetHistamine H1 receptor(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM255474(US9481688, 1 | US9481688, 3)
Affinity DataKi:  20.6nM ΔG°:  -43.9kJ/molepH: 7.6 T: 2°CAssay Description:[3H]-Pyrilamine binding experiments are carried out in SPA (scintillation proximity assay) 96-well format. Membranes used in this assay are prepared ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H1 receptor(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM255474(US9481688, 1 | US9481688, 3)
Affinity DataKi:  58.8nM ΔG°:  -41.3kJ/molepH: 7.6 T: 2°CAssay Description:[3H]-Pyrilamine binding experiments are carried out in SPA (scintillation proximity assay) 96-well format. Membranes used in this assay are prepared ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent