Affinity DataEC50: 200nMAssay Description:Agonist activity at human recombinant histamine H1 receptor expressed in Sf9 cells coexpressing RGS4 by steady-state GTPase activity assayMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataEC50: 2.51E+3nMAssay Description:H1-Histamine receptor agonism on Guinea pig aorta was evaluated (SEM 0.03-0.18)More data for this Ligand-Target Pair