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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM128114'
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbvie

US Patent
LigandPNGBDBM128114(US8796297, 20)
Affinity DataKi:  58.9nM ΔG°:  -38.4kJ/molepH: 7.4 T: 2°CAssay Description:The rat H3 receptor was cloned and expressed in cells, and competition binding assays carried out, according to methods previously described (see Esb...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM128114(US8796297, 20)
Affinity DataKi:  302nM ΔG°:  -34.6kJ/molepH: 7.4 T: 2°CAssay Description:The rat H3 receptor was cloned and expressed in cells, and competition binding assays carried out, according to methods previously described (see Esb...More data for this Ligand-Target Pair
In DepthDetails US Patent