Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM27201'
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM27201(4-{methyl[(1R,2S,5S,6S,9R,12S,13R,16S)-6,7,13-trim...)
Affinity DataKi:  1.66nM ΔG°:  -50.1kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM27201(4-{methyl[(1R,2S,5S,6S,9R,12S,13R,16S)-6,7,13-trim...)
Affinity DataKi:  24nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed