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Found 3 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50050168'
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50050168(3-(4-Iodo-phenyl)-propionic acid 3-(1H-imidazol-4-...)
Affinity DataKi:  47nMAssay Description:In vitro antagonistic activity tested against Histamine H3 receptor on synaptosomes from rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50050168(3-(4-Iodo-phenyl)-propionic acid 3-(1H-imidazol-4-...)
Affinity DataKi:  50nMAssay Description:In vitro antagonistic activity tested against Histamine H3 receptor on synaptosomes from rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50050168(3-(4-Iodo-phenyl)-propionic acid 3-(1H-imidazol-4-...)
Affinity DataKi:  79.4nMAssay Description:Binding affinity towards Histamine H3 receptor on synaptosomes from rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed