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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50051214'
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50051214((4-Fluoro-benzyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  23nMAssay Description:In vitro antagonistic activity of the compound against Histamine H3 receptor on Synaptosomes of rat cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50051214((4-Fluoro-benzyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  25.1nMAssay Description:Binding affinity against Histamine H3 receptor on Synaptosomes from rat cerebral cortex was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed