Affinity DataKi: 1nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 459nMAssay Description:Antagonist activity at recombinant human H3 receptor expressed on CHO-K1 cells assessed as cAMP level by luciferase gene reporter assayMore data for this Ligand-Target Pair