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Found 4 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50217581'
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50217581(4-(4-(1-isopropylpiperidin-4-yloxy)benzyl)morpholi...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50217581(4-(4-(1-isopropylpiperidin-4-yloxy)benzyl)morpholi...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in human SK-N-MC cells after 1 hr by fluid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50217581(4-(4-(1-isopropylpiperidin-4-yloxy)benzyl)morpholi...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50217581(4-(4-(1-isopropylpiperidin-4-yloxy)benzyl)morpholi...)
Affinity DataKi:  2.14nMAssay Description:Mean binding affinity for human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed