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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50297717'
TargetHistamine H3 receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50297717((6-(1-isopropylpiperidin-4-yloxy)naphthalen-2-yl)(...)
Affinity DataKi:  40nMAssay Description:Inhibition of human histamine H3 expressed in CHO cells by saturation binding experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50297717((6-(1-isopropylpiperidin-4-yloxy)naphthalen-2-yl)(...)
Affinity DataEC50:  17nMAssay Description:Inverse agonist activity at human histamine H3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed