Affinity DataKi: 40nMAssay Description:Inhibition of human histamine H3 expressed in CHO cells by saturation binding experimentMore data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Inverse agonist activity at human histamine H3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair