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Found 2 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase KAT2A' and Ligand = 'BDBM50467835'
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50467835(CHEMBL217676)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant human GCN5 using histone peptide as substrate in presence of [14C]-acetyl CoA by microbeta counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50467835(CHEMBL217676)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant human GST-tagged Gcn5 using H3 as substrate in presence of [3H]-acetyl-CoA by phosphor image analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed