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Found 4 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase KAT2B' and Ligand = 'BDBM50398244'
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50398244(CHEMBL609728)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of biotinylated Tat-KAc50 peptide binding to PCAFMore data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50398244(CHEMBL609728)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of biotinylated small molecule ligand from His/FLAG-tagged PCAF bromodomain (719 to 832 residues) (unknown origin) after 15 mins by Alph...More data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50398244(CHEMBL609728)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of biotinylated Tat-AcK50 binding to GST-fused PCAF bromodomain (719 to 832 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50398244(CHEMBL609728)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of GST-tagged PCAF bromodomain (719 to 832 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using Biotin-GISYGR-AcK-KKR...More data for this Ligand-Target Pair